Gassman indole synthesis

Schematic representation of the Gassman indole synthesis.
Mechanism of the Gassman indole synthesis
Mechanism of the Gassman indole synthesis
Original publication
Review
Sample reactions
intermediate structure
Et3N, t-BuOCl, PhNH2
CH2Cl2, MeCN
-45 °C to RT, 3 h, 77%
intermediate structure